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Charles Belunis

Hoffmann-La Roche

19

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1025

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Deconstruction of a Nutlin: Dissecting the Binding Determinants of a Potent Protein–Protein Interaction Inhibitor

2013 ACS Medicinal Chemistry Letters
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Mitogen-activated protein kinase kinase 1 (MEK1) in complex with CH4858061 and MgATP

2011
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Design and synthesis of novel allosteric MEK inhibitor CH4987655 as an orally available anticancer agent.

2011 Bioorganic & Medicinal Chemistry Letters
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Crystal structures of IL-2-inducible T cell kinase complexed with inhibitors: insights into rational drug design and activity regulation.

2010 Chemical Biology & Drug Design
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Fatty acid modulators for the treatment of diabesity

2007 Drug Discovery Today: Therapeutic Strategies
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Protein-protein interactions involved in the recognition of p27 by E3 ubiquitin ligase.

2003 Biochemical Journal
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PEPCK complex with PEP

2002
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Crystal structure of human cytosolic phosphoenolpyruvate carboxykinase reveals a new GTP-binding site.

2002 Journal of Molecular Biology
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PEPCK complex with nonhydrolyzable GTP analog, native data

2002
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Peptide and peptide mimetic inhibitors of antigen presentation by HLA-DR class II MHC molecules. Design, structure-activity relationships, and X-ray crystal structures.

2000 Journal of Medicinal Chemistry
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Citations (89)