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Richard S. Alexander

University of Pennsylvania

30

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1982

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Fragment Binding to β-Secretase 1 without Catalytic Aspartate Interactions Identified via Orthogonal Screening Approaches

2017
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Behandlungsverfahren mit allosterischen verarbeitungshemmern für matrix-metalloproteinasen

2012
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Méthodes de conception, de sélection et/ou d'optimisation d'inhibiteurs de traitement allostériques pour métalloprotéinases matricielles

2012
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Méthodes de traitement utilisant des inhibiteurs de maturation allostériques pour métalloprotéinases matricielles

2012
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Discovery of 1-(4-Methoxyphenyl)-7-oxo-6-(4-(2-oxopiperidin-1-yl)phenyl)-4,5,6,7-tetrahydro- 1H-pyrazolo[3,4-c]pyridine-3-carboxamide (Apixaban, BMS-562247), a Highly Potent, Selective, Efficacious, and Orally Bioavailable Inhibitor of Blood Coagulation Factor Xa.

2007 Journal of Medicinal Chemistry
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Triazolopyridazines as modulators of tyrosine kinases

2006
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Porcine Factor IXa Complexed to 1-{3-[amino(imino)methyl]phenyl}-N-[4-(1H-benzimidazol-1-yl)-2-fluorophenyl]-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide

2005
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Discovery of 1-(3‘-Aminobenzisoxazol-5‘-yl)-3-trifluoromethyl-N-[2-fluoro-4- [(2‘-dimethylaminomethyl)imidazol-1-yl]phenyl]-1H-pyrazole-5-carboxyamide Hydrochloride (Razaxaban), a Highly Potent, Selective, and Orally Bioavailable Factor Xa Inhibitor

2005 Journal of Medicinal Chemistry
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Discovery of 1-(2-Aminomethylphenyl)-3-trifluoromethyl-N-[3-fluoro-2'-(aminosulfonyl)[1,1'-biphenyl)]-1H-pyrazole-5-carboxyamide (DPC602), a Potent, Selective, and Orally Bioavailable Factor Xa Inhibitor.

2003 Journal of Medicinal Chemistry
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Design and synthesis of isoxazoline derivatives as factor Xa inhibitors. 1.

1999 Journal of Medicinal Chemistry
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Citations (88)