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Nicholas Jones
Nicholas Jones
Merck & Co.
Amyloid precursor protein secretase
Pyrazolopyridine
Biochemistry
γ secretase modulator
γ secretase
4
Papers
85
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Antagonism of the adenosine A2A receptor attenuates akathisia-like behavior induced with MP-10 or aripiprazole in a novel non-human primate model
2014
Pharmacology, Biochemistry and Behavior
Carina J. Bleickardt
Tatiana M. Kazdoba
Nicholas Jones
John C. Hunter
Robert Hodgson
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Citations (10)
A2A receptor antagonists do not induce dyskinesias in drug-naive or l-dopa sensitized rats
2013
Brain Research Bulletin
Nicholas Jones
Carina J. Bleickardt
Deborra Mullins
Eric M. Parker
Robert Hodgson
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Citations (22)
Discovery of fused 5,6-bicyclic heterocycles as γ-secretase modulators
2011
Bioorganic & Medicinal Chemistry Letters
Jun Qin
Pawan K. Dhondi
Xianhai Huang
Mihirbaran Mandal
Zhiqiang Zhao
Dmitri Pissarnitski
Wei Zhou
Robert Aslanian
Zhaoning Zhu
William J. Greenlee
John Clader
Lili Zhang
Mary Cohen-Williams
Nicholas Jones
Lynn Hyde
Anandan Palani
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Citations (24)
Discovery of a Potent Pyrazolopyridine Series of γ-Secretase Modulators
2011
ACS Medicinal Chemistry Letters
Jun Qin
Wei Zhou
Xianhai Huang
Pawan K. Dhondi
Anandan Palani
Robert G. Aslanian
Zhaoning Zhu
William J. Greenlee
Mary Cohen-Williams
Nicholas Jones
Lynn A. Hyde
Lili Zhang
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Citations (29)
1