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Jianming Yu
Jianming Yu
Stereochemistry
Chemistry
Philosophy
Pyridine
Molecular biology
4
Papers
17
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0
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Structure-activity relationship studies and discovery of a potent transient receptor potential vanilloid (TRPV1) antagonist 4-[3-chloro-5-[(1S)-1,2-dihydroxyethyl]-2-pyridyl]-N-[5-(trifluoromethyl)-2-pyridyl]-3,6-dihydro-2H-pyridine-1-carboxamide (V116517) as a clinical candidate for pain management.
2014
Journal of Medicinal Chemistry
Laykea Tafesse
Toshiyuki Kanemasa
Noriyuki Kurose
Jianming Yu
Toshiyuki Asaki
Gang Wu
Yuka Iwamoto
Yoshitaka Yamaguchi
Chiyou Ni
John Engel
Naoki Tsuno
Aniket Patel
Xiaoming Zhou
Takuya Shintani
Kevin C. Brown
Tsuyoshi Hasegawa
Manjunath Shet
Yasuyoshi Iso
Akira Kato
Donald J. Kyle
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Citations (17)
Analogues de benzomorphane et leur utilisation
2013
Jeffrey Lockman
Laykea Tafesse
Jiangchao Yao
Jianming Yu
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Composés de type benzomorphane utilisés en tant que modulateurs des récepteurs aux opiacés
2013
Laykea Tafesse
Jae Hyun Park
Jianming Yu
David Rosen
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Composés de pyridine et ses utilisations
2011
Chiyou Ni
Bin Shao
Laykea Tafesse
Jiangchao Yao
Jianming Yu
Xiaoming Zhou
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