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Kevin C. Brown
Kevin C. Brown
Purdue Pharma
Stereochemistry
Chemistry
Ligand
Piperidine
Organic chemistry
5
Papers
33
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Structure-activity relationship studies and discovery of a potent transient receptor potential vanilloid (TRPV1) antagonist 4-[3-chloro-5-[(1S)-1,2-dihydroxyethyl]-2-pyridyl]-N-[5-(trifluoromethyl)-2-pyridyl]-3,6-dihydro-2H-pyridine-1-carboxamide (V116517) as a clinical candidate for pain management.
2014
Journal of Medicinal Chemistry
Laykea Tafesse
Toshiyuki Kanemasa
Noriyuki Kurose
Jianming Yu
Toshiyuki Asaki
Gang Wu
Yuka Iwamoto
Yoshitaka Yamaguchi
Chiyou Ni
John Engel
Naoki Tsuno
Aniket Patel
Xiaoming Zhou
Takuya Shintani
Kevin C. Brown
Tsuyoshi Hasegawa
Manjunath Shet
Yasuyoshi Iso
Akira Kato
Donald J. Kyle
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Heterocyclic substituted piperidines as ORL-1 ligand-
2008
Yoshiyasu Baba
Kevin C. Brown
R. Richard Goehring
Naoki Tsuno
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Composés de pipéridine substituée hétérocycliques et leurs utilisations
2008
Yoshiyasu Baba
Kevin C. Brown
R. Richard Goehring
Naoki Tsuno
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Composés de piperidine substituée heterocycliques comme ligands de ORL-1
2008
Yoshiyasu Baba
Kevin C. Brown
R. Richard Goehring
Naoki Tsuno
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1,3-Dihydro-2,1,3-benzothiadiazol-2,2-diones and 3,4-dihydro-1H-2,1,3-benzothidiazin-2,2-diones as ligands for the NOP receptor.
2004
Bioorganic & Medicinal Chemistry Letters
R. Richard Goehring
John Whitehead
Kevin C. Brown
Khondaker Islam
Xin Wen
Xiaoming Zhou
Zhengming Chen
Kenneth J. Valenzano
Wendy Miller
Shen Shan
Donald J. Kyle
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Citations (16)
1