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Aniket Patel
Aniket Patel
Purdue Pharma
TRPV1
Biochemistry
Organic chemistry
In vivo
Antagonist
3
Papers
63
Citations
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Phenylarsine oxide as a redox modulator of transient receptor potential vanilloid type 1 channel function
2015
Journal of Neuroscience Research
Kevin P. Carlin
Gang Wu
Aniket Patel
Gregg Crumley
Victor I. Ilyin
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Structure-activity relationship studies and discovery of a potent transient receptor potential vanilloid (TRPV1) antagonist 4-[3-chloro-5-[(1S)-1,2-dihydroxyethyl]-2-pyridyl]-N-[5-(trifluoromethyl)-2-pyridyl]-3,6-dihydro-2H-pyridine-1-carboxamide (V116517) as a clinical candidate for pain management.
2014
Journal of Medicinal Chemistry
Laykea Tafesse
Toshiyuki Kanemasa
Noriyuki Kurose
Jianming Yu
Toshiyuki Asaki
Gang Wu
Yuka Iwamoto
Yoshitaka Yamaguchi
Chiyou Ni
John Engel
Naoki Tsuno
Aniket Patel
Xiaoming Zhou
Takuya Shintani
Kevin C. Brown
Tsuyoshi Hasegawa
Manjunath Shet
Yasuyoshi Iso
Akira Kato
Donald J. Kyle
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Citations (17)
4-(2-pyridyl)piperazine-1-carboxamides: potent vanilloid receptor 1 antagonists.
2003
Bioorganic & Medicinal Chemistry Letters
Qun Sun
Laykea Tafesse
Khondaker Islam
Xiaoming Zhou
Sam Victory
Chongwu Zhang
Mohamed Hachicha
Lori Schmid
Aniket Patel
Yakov Rotshteyn
Kenneth J. Valenzano
Donald J. Kyle
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Citations (46)
1