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Claudio Chuaqui

Biogen Idec

44

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Discovery of SY-5609: A Selective, Noncovalent Inhibitor of CDK7.

2021 Journal of Medicinal Chemistry
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Abstract 4421: SY-5609, an orally available selective CDK7 inhibitor demonstrates broad anti-tumor activity in vivo

2019 Cancer Research
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Discovery and Optimization of a Novel Series of Highly Selective JAK1 Kinase Inhibitors

2018 Journal of Medicinal Chemistry
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Discovery of pyrazolo[1,5-a]pyrimidine B-cell lymphoma 6 (BCL6) binders and optimization to high affinity macrocyclic inhibitors

2017 Journal of Medicinal Chemistry
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Utilization of Structure-Based Design to Identify Novel, Irreversible Inhibitors of EGFR Harboring the T790M Mutation

2016 ACS Medicinal Chemistry Letters
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EGFR-K IN COMPLEX WITH N-[3-[[5-chloro-4-(1H-indol-3-yl)pyrimidin-2-yl]amino]-4-methoxy-phenyl] Prop-2-enamide

2013
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Potent and Selective Inhibitors of CK2 Kinase Identified through Structure-Guided Hybridization

2012 ACS Medicinal Chemistry Letters
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Pyrazolone based TGFβR1 kinase inhibitors

2010 Bioorganic & Medicinal Chemistry Letters
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2-Aminoimidazoles inhibitors of TGF-β receptor 1

2009 Bioorganic & Medicinal Chemistry Letters
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SM16, an Orally Active TGF-β Type I Receptor Inhibitor Prevents Myofibroblast Induction and Vascular Fibrosis in the Rat Carotid Injury Model

2008 Arteriosclerosis, Thrombosis, and Vascular Biology
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Citations (70)