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Massimiliano Fonsi

Merck & Co.

13

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402

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Intra Articular (IA) Hyaluronic Acid (HA) and Chondroitin Sulfate (CS): Pharmacokinetic (PK) investigation in rat osteoarthritic model

2019 Current Therapeutic Research-clinical and Experimental
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N-(2-alkylaminoethyl)-4-(1,2,4-oxadiazol-5-yl)piperazine-1-carboxamides as highly potent smoothened antagonists.

2011 Bioorganic & Medicinal Chemistry Letters
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Identification of MK-5710 ((8 aS)-8 a-methyl-1,3-dioxo-2-[(1 S,2 R)-2-phenylcyclopropyl]- N-(1-pheny

2011 International Journal of Food Microbiology
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Discovery of a Potent Class I Selective Ketone Histone Deacetylase Inhibitor with Antitumor Activity in Vivo and Optimized Pharmacokinetic Properties

2009 Journal of Medicinal Chemistry
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Metabolism-related liabilities of a potent histone deacetylase (HDAC) inhibitor and relevance of the route of administration on its metabolic fate

2009 Xenobiotica
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Abstract #1921: Development of MK-4827: a novel oral poly(ADP-ribose)polymerase (PARP) inhibitor efficacious in BRCA-1 and -2 mutant tumors

2009 Cancer Research
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Discovery of 2-{4-[(3S)-piperidin-3-yl]phenyl}-2H-indazole-7-carboxamide (MK-4827): a novel oral poly(ADP-ribose)polymerase (PARP) inhibitor efficacious in BRCA-1 and -2 mutant tumors.

2009 Journal of Medicinal Chemistry
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Design and synthesis of bicyclic pyrimidinones as potent and orally bioavailable HIV-1 integrase inhibitors.

2008 Journal of Medicinal Chemistry
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Optimization of a series of potent and selective ketone histone deacetylase inhibitors.

2008 Bioorganic & Medicinal Chemistry Letters
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High-Throughput Microsomal Stability Assay for Screening New Chemical Entities in Drug Discovery

2008 Journal of Biomolecular Screening
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Citations (26)