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Mitsuru Sasaki
Mitsuru Sasaki
Takeda Pharmaceutical Company
Stereochemistry
Chemistry
Biochemistry
Urinary bladder
Chemical synthesis
3
Papers
45
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Identification of 3-aminomethyl-1,2-dihydro-4-phenyl-1-isoquinolones: A new class of potent, selective, and orally active non-peptide dipeptidyl peptidase IV inhibitors that form a unique interaction with Lys554
2011
Bioorganic & Medicinal Chemistry
Yoshihiro Banno
Yasufumi Miyamoto
Mitsuru Sasaki
Satoru Oi
Tomoko Asakawa
Osamu Kataoka
Koji Takeuchi
Nobuhiro Suzuki
Koji Ikedo
Takuo Kosaka
Shigetoshi Tsubotani
Akiyoshi Tani
Miyuki Funami
Michiko Tawada
Yoshio Yamamoto
Kathleen Aertgeerts
Jason Yano
Hironobu Maezaki
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Citations (31)
Novel acetylcholinesterase inhibitor as increasing agent on rhythmic bladder contractions: SAR of 8-{3-[1-(3-fluorobenzyl)piperidin-4-yl]propanoyl}-1,2,5,6-tetrahydro-4H-pyrrolo[3,2,1-ij]quinolin-4-one (TAK-802) and related compounds
2005
Bioorganic & Medicinal Chemistry
Yuji Ishichi
Mitsuru Sasaki
Masaki Setoh
Tetsuya Tsukamoto
Seiji Miwatashi
Hiroshi Nagabukuro
Satoshi Okanishi
Shigemitsu Imai
Reiko Saikawa
Takayuki Doi
Yuji Ishihara
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Citations (14)
Composes azotes hererocycliques condenses; procede de fabrication et agents les renfermant
1999
Yuji Ishihara
Yukio Fujisawa
Naoki Furuyama
Yuji Ishichi
Mitsuru Sasaki
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