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Frédéric Ausseil

Centre national de la recherche scientifique

35

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Identification of a novel quinoline-based DNA demethylating compound highly potent in cancer cells

2019 Clinical Epigenetics
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Rational Design of Bisubstrate-Type Analogues as Inhibitors of DNA Methyltransferases in Cancer Cells

2017 Journal of Medicinal Chemistry
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Chapter 3 – Drug Discovery Methods

2016
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Identification and optimization of hydrazone-gallate derivatives as specific inhibitors of DNA methyltransferase 3A

2016 Future Medicinal Chemistry
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Asymmetric Synthesis and Binding Study of New Long‐Chain HPA‐12 Analogues as Potent Ligands of the Ceramide Transfer Protein CERT

2016 Chemistry: A European Journal
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Design and synthesis of new non nucleoside inhibitors of DNMT3A.

2015 Bioorganic & Medicinal Chemistry
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The CERT antagonist HPA-12: first practical synthesis and individual binding evaluation of the four stereoisomers.

2015 Bioorganic & Medicinal Chemistry
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New insights on the mechanism of quinoline-based DNA methyltransferase inhibitors

2015 Journal of Biological Chemistry
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Development of a CERT START Domain–Ceramide HTRF Binding Assay and Application to Pharmacological Studies and Screening

2015 Journal of Biomolecular Screening
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Properly Substituted Analogues of BIX-01294 Lose Inhibition of G9a Histone Methyltransferase and Gain Selective Anti-DNA Methyltransferase 3A Activity

2014 PLOS ONE
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Citations (28)