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Akinola Soyode-Johnson
Akinola Soyode-Johnson
Johnson & Johnson Pharmaceutical Research and Development
Chemistry
Stereochemistry
Trifluoromethyl
Organic chemistry
Pyridine
5
Papers
59
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Design, Synthesis and Preclinical Evaluation of 3-Methyl-6-(5-thiophenyl)-1,3-dihydro-imidazo[4,5-b]pyridin-2-ones as Selective GluN2B Negative Allosteric Modulators for the Treatment of Mood Disorders
2020
Journal of Medicinal Chemistry
Christa C. Chrovian
Akinola Soyode-Johnson
Brice Stenne
Daniel J. Pippel
Jeffrey Schoellerman
Brian Lord
Alexandra S Needham
Chunfang Xia
Kevin J. Coe
Kia Sepassi
Freddy Schoetens
Brian Scott
Leslie Nguyen
Xiaohui Jiang
Tatiana Koudriakova
Bartosz Balana
Michael A. Letavic
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Citations (2)
A Dipolar Cycloaddition Reaction To Access 6-Methyl-4,5,6,7-tetrahydro-1H-[1,2,3]triazolo[4,5-c]pyridines Enables the Discovery Synthesis and Preclinical Profiling of a P2X7 Antagonist Clinical Candidate
2018
Journal of Medicinal Chemistry
Christa C. Chrovian
Akinola Soyode-Johnson
Alexander A. Peterson
Christine Gelin
Xiaohu Deng
Curt A. Dvorak
Nicholas I. Carruthers
Brian Lord
Ian Fraser
Leah Aluisio
Kevin J. Coe
Brian Scott
Tatiana Koudriakova
Freddy Schoetens
Kia Sepassi
David Gallacher
Anindya Bhattacharya
Michael A. Letavic
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Citations (34)
Novel Phenyl-Substituted 5,6-Dihydro-[1,2,4]triazolo[4,3-a]pyrazine P2X7 Antagonists with Robust Target Engagement in Rat Brain
2016
ACS Chemical Neuroscience
Christa C. Chrovian
Akinola Soyode-Johnson
Hong Ao
Genesis M. Bacani
Nicholas I. Carruthers
Brian Lord
Leslie Nguyen
Jason C. Rech
Qi Wang
Anindya Bhattacharya
Michael A. Letavic
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Citations (18)
Octahydropyrrolo[3,4-c]pyrroles disubstitués en tant que modulateurs de récepteur d'orexine
2010
Wenying Chai
Michael A. Letavic
Kiev S. Ly
Daniel J. Pippel
Dale A. Rudolph
Kathleen C. Sappey
Brad M. Savall
Chandravadan R. Shah
Brock T. Shireman
Akinola Soyode-Johnson
Emily M. Stocking
Devin M. Swanson
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Novel substituted pyrrolidines are high affinity histamine H3 receptor antagonists
2010
Bioorganic & Medicinal Chemistry Letters
Emily M. Stocking
Leah Aluisio
John R. Atack
Pascal Bonaventure
Nicholas I. Carruthers
Christine Dugovic
Anita Everson
Ian C. Fraser
Xiaohui Jiang
Perry Leung
Brian Lord
Kiev S. Ly
Kirsten L. Morton
Diane Nepomuceno
Chandravadan R. Shah
Jonathan Shelton
Akinola Soyode-Johnson
Michael A. Letavic
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Citations (5)
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