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Hiroshi Nakamura
Hiroshi Nakamura
Pfizer
Chemistry
Structure–activity relationship
Agonist
Anxiolytic
Nociceptin receptor
4
Papers
73
Citations
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Discovery of 1‐[1‐(1‐Methylcyclooctyl)‐4‐piperidinyl]‐2‐[(3R)‐3‐piperidinyl]‐1H‐benzimidazole: Integrated Drug‐Design and Structure–Activity Relationships for Orally Potent, Metabolically Stable and Potential‐Risk Reduced Novel Non‐Peptide Nociceptin/Orphanin FQ Receptor Agonist as Antianxiety Drug‡
2009
Chemical Biology & Drug Design
Shigeo Hayashi
Akiko Hirao
Hiroshi Nakamura
Kenzo Yamamura
Kunihiko Mizuno
Hiroyo Yamashita
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Citations (12)
Novel Non-Peptide Nociceptin/Orphanin FQ Receptor Agonist, 1-[1-(1-Methylcyclooctyl)-4-piperidinyl]-2-[(3R)-3-piperidinyl]-1H-benzimidazole: Design, Synthesis, and Structure−Activity Relationship of Oral Receptor Occupancy in the Brain for Orally Potent Antianxiety Drug(1, 2)
2009
Journal of Medicinal Chemistry
Shigeo Hayashi
Akiko Hirao
Aki Imai
Hiroshi Nakamura
Yoshinori Murata
Katsuyo Ohashi
Eriko Nakata
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Discovery of (-)-6-[2-[4-(3-fluorophenyl)-4-hydroxy-1-piperidinyl]-1-hydroxyethyl]-3,4-dihydro-2(1H)-quinolinone--a potent NR2B-selective N-methyl D-aspartate (NMDA) antagonist for the treatment of pain.
2007
Bioorganic & Medicinal Chemistry Letters
Makoto Kawai
Kazuo Ando
Yukari Matsumoto
Isao Sakurada
Masako Hirota
Hiroshi Nakamura
Atsuko Ohta
Masaki Sudo
Kazunari Hattori
Tadashi Takashima
Masanori Hizue
Shuzo Watanabe
Isami Fujita
Mayumi Mizutani
Mitsuhiro Kawamura
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Discovery of novel and orally active NR2B-selective N-methyl-D-aspartate (NMDA) antagonists, pyridinol derivatives with reduced HERG binding affinity.
2007
Bioorganic & Medicinal Chemistry Letters
Makoto Kawai
Hiroshi Nakamura
Isao Sakurada
Hirohisa Shimokawa
Hirotaka Tanaka
Miyako Matsumizu
Kazuo Ando
Kazunari Hattori
Atsuko Ohta
Seiji Nukui
Atsushi Omura
Mitsuhiro Kawamura
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Citations (12)
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