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Isao Sakurada
Isao Sakurada
Pfizer
Chemistry
Stereochemistry
Organic chemistry
Biochemistry
Antagonist
5
Papers
58
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Discovery of (-)-6-[2-[4-(3-fluorophenyl)-4-hydroxy-1-piperidinyl]-1-hydroxyethyl]-3,4-dihydro-2(1H)-quinolinone--a potent NR2B-selective N-methyl D-aspartate (NMDA) antagonist for the treatment of pain.
2007
Bioorganic & Medicinal Chemistry Letters
Makoto Kawai
Kazuo Ando
Yukari Matsumoto
Isao Sakurada
Masako Hirota
Hiroshi Nakamura
Atsuko Ohta
Masaki Sudo
Kazunari Hattori
Tadashi Takashima
Masanori Hizue
Shuzo Watanabe
Isami Fujita
Mayumi Mizutani
Mitsuhiro Kawamura
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Discovery of novel and orally active NR2B-selective N-methyl-D-aspartate (NMDA) antagonists, pyridinol derivatives with reduced HERG binding affinity.
2007
Bioorganic & Medicinal Chemistry Letters
Makoto Kawai
Hiroshi Nakamura
Isao Sakurada
Hirohisa Shimokawa
Hirotaka Tanaka
Miyako Matsumizu
Kazuo Ando
Kazunari Hattori
Atsuko Ohta
Seiji Nukui
Atsushi Omura
Mitsuhiro Kawamura
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Structure–activity relationship study of novel NR2B-selective antagonists with arylamides to avoid reactive metabolites formation
2007
Bioorganic & Medicinal Chemistry Letters
Makoto Kawai
Isao Sakurada
Asato Morita
Yuko Iwamuro
Kazuo Ando
Hirofumi Omura
Sachiko Sakakibara
Tsutomu Masuda
Hiroki Koike
Teruki Honma
Kazunari Hattori
Tadayuki Takashima
Kunihiko Mizuno
Mayumi Mizutani
Mitsuhiro Kawamura
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Citations (9)
Derives d'amide therapeutiques
2005
Makoto Kawai
Mitsuhiro Kawamura
Isao Sakurada
Asato Morita
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Direct Chlorohydrin and Acetoxy Alcohol Synthesis from Olefins Promoted by a Lewis Acid, Bis(trimethylsilyl) Peroxide and (CH3)3SiX
2000
Journal of the American Chemical Society
Isao Sakurada
Shingo Yamasaki
Richard Göttlich
Takehiko Iida
and Motomu Kanai
Masakatsu Shibasaki
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Citations (27)
1