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Xiaofei Liang
Xiaofei Liang
Hefei Institutes of Physical Science
Chemistry
In vivo
Kinase
Phosphorylation
IC50
7
Papers
26
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Discovery of IHMT-EZH2-115 as a Potent and Selective Enhancer of Zeste Homolog 2 (EZH2) Inhibitor for the Treatment of B-Cell Lymphomas.
2021
Journal of Medicinal Chemistry
Bin Zhou
Xiaofei Liang
Husheng Mei
Qi Shuang
Zongru Jiang
Aoli Wang
Fengming Zou
Qingwang Liu
Juan Liu
Wenliang Wang
Chen Hu
Yongfei Chen
Zuowei Wang
Beilei Wang
Li Wang
Jing Liu
Qingsong Liu
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An ultra-long circulating nanoparticle for reviving a highly selective BCR-ABL inhibitor in long-term effective and safe treatment of chronic myeloid leukemia
2020
Nanomedicine: Nanotechnology, Biology and Medicine
Liyi Fu
Fengming Zou
Qingwang Liu
Beilei Wang
Junqing Wang
Huamin Liang
Xiaofei Liang
Jing Liu
Jinjun Shi
Qingsong Liu
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Discovery of (S)-2-(1-(4-Amino-3-(3-fluoro-4-methoxyphenyl)-1H-pyrazolo[3,4-d]pyrimidin-1-yl)propyl)-3-cyclopropyl-5-fluoroquinazolin-4(3H)-one (IHMT-PI3Kδ-372) as a Potent and Selective PI3Kδ Inhibitor for the Treatment of Chronic Obstructive Pulmonary Disease.
2020
Journal of Medicinal Chemistry
Li Feng
Xiaofei Liang
Zongru Jiang
Aoli Wang
Wang Junjie
Cheng Chen
Wenliang Wang
Fengming Zou
Ziping Qi
Qingwang Liu
Zhenquan Hu
Jiangyan Cao
Hong Wu
Beilei Wang
Li Wang
Jing Liu
Qingsong Liu
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Discovery of 6'-chloro-N-methyl-5'-(phenylsulfonamido)-[3,3'-bipyridine]-5-carboxamide (CHMFL-PI4K-127) as a novel Plasmodium falciparum PI(4)K inhibitor with potent antimalarial activity against both blood and liver stages of Plasmodium.
2020
European Journal of Medicinal Chemistry
Xiaofei Liang
Zongru Jiang
Zhenghui Huang
Feng Li
Cheng Chen
Chen Hu
Wenliang Wang
Zhenquan Hu
Qingwang Liu
Beilei Wang
Li Wang
Ziping Qi
Jing Liu
Lubin Jiang
Qingsong Liu
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Discovery of N-(4-(6-Acetamidopyrimidin-4-yloxy)phenyl)-2-(2-(trifluoromethyl)phenyl)acetamide (CHMFL-FLT3-335) as a Potent FMS-like Tyrosine Kinase 3 Internal Tandem Duplication (FLT3-ITD) Mutant Selective Inhibitor for Acute Myeloid Leukemia
2019
Journal of Medicinal Chemistry
Xiaofei Liang
Beilei Wang
Cheng Chen
Aoli Wang
Chen Hu
Fengming Zou
Kailin Yu
Qingwang Liu
Feng Li
Zhenquan Hu
Tingting Lu
Junjie Wang
Li Wang
Ellen Weisberg
Lili Li
Ruixiang Xia
Wenchao Wang
Tao Ren
Jian Ge
Jing Liu
Qingsong Liu
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Citations (12)
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