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Wang Junjie
Wang Junjie
Hefei Institutes of Physical Science
In vivo
Chemistry
Kinome
Kinase
Molecular biology
2
Papers
4
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0
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Discovery of (S)-2-(1-(4-Amino-3-(3-fluoro-4-methoxyphenyl)-1H-pyrazolo[3,4-d]pyrimidin-1-yl)propyl)-3-cyclopropyl-5-fluoroquinazolin-4(3H)-one (IHMT-PI3Kδ-372) as a Potent and Selective PI3Kδ Inhibitor for the Treatment of Chronic Obstructive Pulmonary Disease.
2020
Journal of Medicinal Chemistry
Li Feng
Xiaofei Liang
Zongru Jiang
Aoli Wang
Wang Junjie
Cheng Chen
Wenliang Wang
Fengming Zou
Ziping Qi
Qingwang Liu
Zhenquan Hu
Jiangyan Cao
Hong Wu
Beilei Wang
Li Wang
Jing Liu
Qingsong Liu
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Discovery of (E)-N-(4-methyl-5-(3-(2-(pyridin-2-yl)vinyl)-1H-indazol-6-yl)thiazol-2-yl)-2-(4-methylpiperazin-1-yl)acetamide (IHMT-TRK-284) as a Novel Orally Available Type II TRK Kinase Inhibitor Capable of Overcoming Multiple Resistant Mutants
2020
European Journal of Medicinal Chemistry
Beilei Wang
Wentao Zhang
Xuesong Liu
Fengming Zou
Wang Junjie
Qingwang Liu
Aoli Wang
Zhenquan Hu
Yongfei Chen
Shuang Qi
Zongru Jiang
Cheng Chen
Chen Hu
Wang Li
Wenchao Wang
Qingsong Liu
Jing Liu
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