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Ziping Qi
Ziping Qi
Hefei Institutes of Physical Science
Biochemistry
Kinase
Cancer research
In vivo
Biology
8
Papers
49
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Discovery of 6'-chloro-N-methyl-5'-(phenylsulfonamido)-[3,3'-bipyridine]-5-carboxamide (CHMFL-PI4K-127) as a novel Plasmodium falciparum PI(4)K inhibitor with potent antimalarial activity against both blood and liver stages of Plasmodium.
2020
European Journal of Medicinal Chemistry
Xiaofei Liang
Zongru Jiang
Zhenghui Huang
Feng Li
Cheng Chen
Chen Hu
Wenliang Wang
Zhenquan Hu
Qingwang Liu
Beilei Wang
Li Wang
Ziping Qi
Jing Liu
Lubin Jiang
Qingsong Liu
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Citations (5)
Discovery of a highly potent and selective Bruton's tyrosine kinase inhibitor avoiding impairment of ADCC effects for B-cell non-Hodgkin lymphoma.
2020
Signal Transduction and Targeted Therapy
Juan Liu
Qianmao Liang
Aoli Wang
Fengming Zou
Ziping Qi
Kailin Yu
Qingwang Liu
Cheng Chen
Jing Liu
Qingsong Liu
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Discovery of a Highly Selective VEGFR2 Kinase Inhibitor CHMFL-VEGFR2-002 as a Novel Anti-angiogenesis Agent
2019
Acta Pharmaceutica Sinica B
Zongru Jiang
Li Wang
Xuesong Liu
Cheng Chen
Beilei Wang
Wenliang Wang
Chen Hu
Kailin Yu
Ziping Qi
Qingwang Liu
Aoli Wang
Jing Liu
Guangchen Hong
Wenchao Wang
Qingsong Liu
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Discovery of 2-(4-chloro-3-(trifluoromethyl)phenyl)-N-(4-((6,7-dimethoxyquinolin-4-yl)oxy)phenyl)acetamide (CHMFL-KIT-64) as a Novel Orally Available Potent Inhibitor against Broad Spectrum Mutants of c-KIT Kinase for Gastrointestinal Stromal Tumors (GISTs)
2019
Journal of Medicinal Chemistry
Yun Wu
Beilei Wang
Junjie Wang
Shuang Qi
Fengming Zou
Ziping Qi
Feiyang Liu
Qingwang Liu
Cheng Chen
Chen Hu
Zhenquan Hu
Aoli Wang
Li Wang
Wenchao Wang
Tao Ren
Yujiao Cai
Mingfeng Bai
Qingsong Liu
Jing Liu
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Citations (9)
Discovery of a novel and highly selective CDK9 kinase inhibitor (JSH-009) with potent antitumor efficacy in preclinical acute myeloid leukemia models
2019
Investigational New Drugs
Li Wang
Chen Hu
Aoli Wang
Cheng Chen
Jiaxin Wu
Zongru Jiang
Fengming Zou
Kailin Yu
Hong Wu
Juan Liu
Wenliang Wang
Zuo-wei Wang
Beilei Wang
Ziping Qi
Qingwang Liu
Wenchao Wang
Lili Li
Jian Ge
Jing Liu
Qingsong Liu
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Citations (3)
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