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Darren Mark Le Grand
Darren Mark Le Grand
Novartis
Chemistry
Biochemistry
In vivo
Organic chemistry
Thrombin
11
Papers
70
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Development of autotaxin inhibitors: A series of zinc binding triazoles
2018
Bioorganic & Medicinal Chemistry Letters
Christopher Thomson
Darren Mark Le Grand
Mark R. Dowling
Cara E. Brocklehurst
Colin Chinn
Lucy Elphick
Michael Faller
Mark S. Freeman
Vikki Furminger
Cornelia Gasser
Ahmed Hamadi
Elizabeth Hardaker
Victoria Head
Johan C. Hill
Diana Janus
David William Pearce
Anne-Sophie Poulaud
Emily Stanley
Lilya Sviridenko
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Derivatives of purina as inhibitors of the protein quinasa of tirosina syk.
2000
Stephen Paul Collingwood
Judy Hayler
Darren Mark Le Grand
Henri Mattes
Keith Allan Menear
Clive Victor Walker
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Purine derivative inhibitors of protein kinase syk-tyrosi
2000
Xiaoling Cockcroft
Stephen Paul Collingwood
Judy East Grinstead Hayler
Darren Mark Le Grand
Henri Mattes
Keith Allan Menear
Clive Victor Walker
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Studies towards the identification of potent, selective and bioavailable thrombin inhibitors.
1999
Bioorganic & Medicinal Chemistry Letters
John Ambler
Emma Baker
Dave Bentley
Lyndon Nigel Brown
Keith Butler
Paul Butler
Dave Farr
Karen Dunnet
Darren Mark Le Grand
Judy Hayler
Diana Janus
Darryl Brynley Jones
Keith Menear
Mark Mercer
Garrick Smith
Mark Talbot
Morris Tweed
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Citations (7)
The discovery of orally available thrombin inhibitors: optimisation of the P1 pharmacophore.
1999
Bioorganic & Medicinal Chemistry Letters
John Ambler
David Bentley
Lyndon Nigel Brown
Karen Dunnet
Dave Farr
Diana Janus
Darren Mark Le Grand
Keith Menear
Mark Mercer
Mark Talbot
Morris Tweed
Bernard Wathey
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Citations (6)
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