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Osamu Kubo
Osamu Kubo
Takeda Pharmaceutical Company
Stereochemistry
Chemistry
Trifluoromethyl
Biochemistry
Potency
5
Papers
34
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Discovery of a Novel Series of Indolinylpyrimidine-based GPR119 Agonists: Elimination of Ether-a-go-go-related Gene Liability Using a Hydrogen Bond acceptor-Focused Approach
2021
Bioorganic & Medicinal Chemistry
Masahiro Kamaura
Osamu Kubo
Hiromichi Sugimoto
Naoyoshi Noguchi
Hirohisa Miyashita
Shin-Ichi Abe
Kae Matsuda
Yoshiyuki Tsujihata
Tomoyuki Odani
Shinji Iwasaki
Toshiki Murata
Kenjiro Sato
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Discovery of a novel series of GPR119 agonists: Design, synthesis, and biological evaluation of N-(Piperidin-4-yl)-N-(trifluoromethyl)pyrimidin-4-amine derivatives.
2021
Bioorganic & Medicinal Chemistry
Osamu Kubo
Kazuaki Takami
Masahiro Kamaura
Koji Watanabe
Hirohisa Miyashita
Shin-Ichi Abe
Kae Matsuda
Yoshiyuki Tsujihata
Tomoyuki Odani
Shinji Iwasaki
Tomoyuki Kitazaki
Toshiki Murata
Kenjiro Sato
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Discovery of a Novel Series of N-Phenylindoline-5-sulfonamide Derivatives as Potent, Selective, and Orally Bioavailable Acyl CoA:Monoacylglycerol Acyltransferase-2 Inhibitors
2015
Journal of Medicinal Chemistry
Kenjiro Sato
Hiroki Takahagi
Takeshi Yoshikawa
Shinji Morimoto
Takafumi Takai
Kousuke Hidaka
Masahiro Kamaura
Osamu Kubo
Ryutaro Adachi
Tsuyoshi Ishii
Toshiyuki Maki
Taisuke Mochida
Shiro Takekawa
Masanori Nakakariya
Nobuyuki Amano
Tomoyuki Kitazaki
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Optimization of a novel series of N-phenylindoline-5-sulfonamide-based acyl CoA:monoacylglycerol acyltransferase-2 inhibitors: Mitigation of CYP3A4 time-dependent inhibition and phototoxic liabilities
2015
Bioorganic & Medicinal Chemistry
Kenjiro Sato
Hiroki Takahagi
Osamu Kubo
Kousuke Hidaka
Takeshi Yoshikawa
Masahiro Kamaura
Masanori Nakakariya
Nobuyuki Amano
Ryutaro Adachi
Toshiyuki Maki
Kazumi Take
Shiro Takekawa
Tomoyuki Kitazaki
Tsuyoshi Maekawa
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Citations (8)
Composé spiro et son utilisation
2008
Takahiko Taniguchi
Kenichi Miyata
Osamu Kubo
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