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Tim Harper
Tim Harper
Bristol-Myers Squibb
Potency
Organic chemistry
Chemistry
hERG
Selectivity
2
Papers
24
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Neutral macrocyclic factor VIIa inhibitors.
2017
Bioorganic & Medicinal Chemistry Letters
Nicholas R. Wurtz
Brandon Parkhurst
Indawati DeLucca
Peter W. Glunz
Wen Jiang
Xiaojun Zhang
Daniel L. Cheney
Jeffrey M. Bozarth
Alan R. Rendina
Anzhi Wei
Tim Harper
Joseph M. Luettgen
Yiming Wu
Pancras C. Wong
Dietmar A. Seiffert
Ruth R. Wexler
E. Scott Priestley
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Citations (5)
Discovery of ((S)-5-(Methoxymethyl)-7-(1-methyl-1H-indol-2-yl)-2-(trifluoromethyl)-4,7-dihydropyrazolo[1,5-a]pyrimidin-6-yl)((S)-2-(3-methylisoxazol-5-yl)pyrrolidin-1-yl)methanone As a Potent and Selective IKur Inhibitor
2012
Journal of Medicinal Chemistry
Heather Finlay
John Lloyd
Wayne Vaccaro
Alexander Kover
Lin Yan
Gauri Bhave
Joseph Prol
Tram N. Huynh
Rao S. Bhandaru
Yolanda Caringal
John D. Dimarco
Jinping Gan
Tim Harper
Christine Huang
Mary Lee Conder
Huabin Sun
Paul Levesque
Michael A. Blanar
Karnail S. Atwal
Ruth R. Wexler
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Citations (19)
1