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Joseph Prol
Joseph Prol
Bristol-Myers Squibb
Potency
Stereochemistry
Chemistry
hERG
Selectivity
2
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54
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Discovery of ((S)-5-(Methoxymethyl)-7-(1-methyl-1H-indol-2-yl)-2-(trifluoromethyl)-4,7-dihydropyrazolo[1,5-a]pyrimidin-6-yl)((S)-2-(3-methylisoxazol-5-yl)pyrrolidin-1-yl)methanone As a Potent and Selective IKur Inhibitor
2012
Journal of Medicinal Chemistry
Heather Finlay
John Lloyd
Wayne Vaccaro
Alexander Kover
Lin Yan
Gauri Bhave
Joseph Prol
Tram N. Huynh
Rao S. Bhandaru
Yolanda Caringal
John D. Dimarco
Jinping Gan
Tim Harper
Christine Huang
Mary Lee Conder
Huabin Sun
Paul Levesque
Michael A. Blanar
Karnail S. Atwal
Ruth R. Wexler
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Citations (19)
Dihydropyrazolopyrimidines containing benzimidazoles as KV1.5 potassium channel antagonists
2009
Bioorganic & Medicinal Chemistry Letters
John Lloyd
Heather Finlay
Karnail S. Atwal
Alexander Kover
Joseph Prol
Lin Yan
Rao S. Bhandaru
Wayne Vaccaro
Tram Huynh
Christine Huang
MaryLee Conder
Tonya Jenkins-West
Huabin Sun
Danshi Li
Paul Levesque
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Citations (35)
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