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Ralph P. Robinson

Pfizer

65

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1442

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Recent Applications of Covalent Chemical Probes for Investigating Drug Off-Target Engagement

2019
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Identification of N-{cis-3-[Methyl(7H-pyrrolo[2,3-d]pyrimidin-4-yl)amino]cyclobutyl}propane-1-sulfonamide (PF-04965842): A Selective JAK1 Clinical Candidate for the Treatment of Autoimmune Diseases.

2018 Journal of Medicinal Chemistry
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Covalent Enzyme Inhibition through Fluorosulfate Modification of a Noncatalytic Serine Residue

2017 ACS Chemical Biology
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Modern Advances in Heterocyclic Chemistry in Drug Discovery

2016 ChemInform
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Visible‐Light‐Driven Photocatalytic Initiation of Radical Thiol—Ene Reactions Using Bismuth Oxide.

2016 ChemInform
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Rational Targeting of Active-Site Tyrosine Residues Using Sulfonyl Fluoride Probes

2015 ACS Chemical Biology
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Facile Synthesis of 2,4-Disubstituted Thiooxazoles and 2,4-Disubstituted Oxazole Sulfonyl Chlorides via Acyl Isothiocyanates and TMS-Diazomethane

2015 Synlett
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A library approach to rapidly discover photoaffinity probes of the mRNA decapping scavenger enzyme DcpS

2015 Molecular BioSystems
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2-Aryl-3-methyloctahydrophenanthrene-2,3,7-triols as Potent Dissociated Glucocorticoid Receptor Agonists

2015 Journal of Medicinal Chemistry
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Visible-Light-Driven Photocatalytic Initiation of Radical Thiol–Ene Reactions Using Bismuth Oxide

2015 Organic Letters
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