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Pauline Kerdoncuff
Pauline Kerdoncuff
Biology
Immunology
Protein kinase A
Cancer
Phosphorylation
4
Papers
89
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Synthesis and SAR of inhibitors of protein kinase CK2: Novel tricyclic quinoline analogs
2012
Bioorganic & Medicinal Chemistry Letters
Mustapha Haddach
Fabrice Pierre
Collin Regan
Cosmin Borsan
Jerome Michaux
Eric Stefan
Pauline Kerdoncuff
Michael Schwaebe
Peter C. Chua
Adam Siddiqui-Jain
Diwata Macalino
Denis Drygin
Sean E. O’Brien
William G. Rice
David M. Ryckman
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Citations (14)
Discovery of CX-5461, the First Direct and Selective Inhibitor of RNA Polymerase I, for Cancer Therapeutics
2012
ACS Medicinal Chemistry Letters
Mustapha Haddach
Michael K. Schwaebe
Jerome Michaux
Johnny Y. Nagasawa
Sean OBrien
Jeffrey P. Whitten
Fabrice Pierre
Pauline Kerdoncuff
Levan Darjania
Ryan Stansfield
Denis Drygin
Kenna Anderes
Chris Proffitt
Josh Bliesath
Adam Siddiqui-Jain
May Omori
Nanni Huser
William G. Rice
David M. Ryckman
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Citations (74)
Abstract A246: Discovery of selective small molecule Pan‐Pim kinase inhibitors with potent oral efficacy in murine xenograft models
2009
Molecular Cancer Therapeutics
Sean OBrien
Mustapha Haddach
Cosmin Borsan
Jerome Michaux
Pauline Kerdoncuff
Michael Schwaebe
Fabrice Pierre
Eric Stefan
Anne‐Sophie Nedellec
Adam Siddiqui-Jain
Nicole Streiner
Diwata Macalino
Denis Drygin
Caroline Ho
Josh Bliesath
May Omori
Ryan Stansfield
Jennifer Phung
David M. Ryckman
William G. Rice
Kenna Anderes
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Discovery of Selective Small Molecule Pan-Pim Kinase Inhibitors with Potent Oral Efficacy in Murine Xenograft Models.
2009
Blood
Sean OBrien
Mustapha Haddach
Cosmin Borsan
Jerome Michaux
Pauline Kerdoncuff
Mike Schwaebe
Fabrice Pierre
Eric Stefan
Anne Sophie Nedellec
Adam Siddiqui-Jain
Nicole Streiner
Diwata Macalino
Denis Drygin
Caroline Ho
Josh Bliesath
May Omori
Ryan Stansfield
Jennifer Phung
David M. Ryckman
William G. Rice
Kenna Anderes
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