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Vivekananda M. Vrudhula

Bristol-Myers Squibb

35

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Design, synthesis and evaluation of constrained tetrahydroimidazopyrimidine derivatives as antagonists of corticotropin-releasing factor type 1 receptor (CRF1R).

2010 Bioorganic & Medicinal Chemistry Letters
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Discovery of 6-chloro-2-trifluoromethyl-7-aryl-7H-imidazo[1,2-a]imidazol-3-ylmethylamines, a novel class of corticotropin-releasing factor receptor type 1 (CRF1R) antagonists

2010 Bioorganic & Medicinal Chemistry Letters
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A strategy to minimize reactive metabolite formation: discovery of (S)-4-(1-cyclopropyl-2-methoxyethyl)-6-[6-(difluoromethoxy)-2,5-dimethylpyridin-3-ylamino]-5-oxo-4,5-dihydropyrazine-2-carbonitrile as a potent, orally bioavailable corticotropin-releasing factor-1 receptor antagonist.

2009 Journal of Medicinal Chemistry
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Separation of maxi-K channel opening 3-substitued-4-arylquinolinone atropisomers by enantioselective supercritical fluid chromatography

2008 Journal of Pharmaceutical and Biomedical Analysis
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Composes de promedicament de pyrrolotriazine aniline utiles en tant qu'inhibiteurs de la kinase

2007
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Analogues (Ib)-(Ic) of a Potent Maxi-K Potassium Channel Opener (Ia) with an Improved Inhibitory Profile Toward Cytochrome P450 Isozymes.

2005 ChemInform
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Reductively Activated Disulfide Prodrugs of Paclitaxel.

2003 ChemInform
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Cephalosporin prodrugs of paclitaxel for immunologically specific activation by L-49-sFv-β-Lactamase fusion protein

2003 Bioorganic & Medicinal Chemistry Letters
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2-Aryl-2,2-difluoroacetamide FKBP12 ligands: synthesis and X-ray structural studies.

2001 Organic Letters
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Comparison of recombinant and synthetically formed monoclonal antibody-beta-lactamase conjugates for anticancer prodrug activation.

1999 Bioconjugate Chemistry
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Citations (19)