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Conrad E. Raab

Merck & Co.

44

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976

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Integrating the Impact of Lipophilicity on Potency and Pharmacokinetic Parameters Enables the Use of Diverse Chemical Space during Small Molecule Drug Optimization.

2020 Journal of Medicinal Chemistry
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Quantitation of Physiological and Biochemical Barriers to siRNA Liver Delivery via Lipid Nanoparticle Platform

2014 Molecular Pharmaceutics
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Remote Electronic Control in the Regioselective Reduction of Succinimides: A Practical, Scalable Synthesis of EP4 Antagonist MF-310

2009 Journal of Organic Chemistry
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Discovery of N-{N-[(3-cyanophenyl)sulfonyl]-4(R)-cyclobutylamino-(L)-prolyl}-4-[(3',5'-dichloroisonicotinoyl) amino]-(L)-phenylalanine (MK-0668), an extremely potent and orally active antagonist of very late antigen-4.

2009 Journal of Medicinal Chemistry
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CYP2C75-Involved Autoinduction of Metabolism in Rhesus Monkeys of MK-0686, a Bradykinin B1 Receptor Antagonist

2008 Journal of Pharmacology and Experimental Therapeutics
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CYP2C75-Involved Autoinduction of Metabolism in Rhesus Monkeys of Methyl 3-Chloro-3′-fluoro-4′-{(1R)-1-[({1-[(trifluoroacetyl)amino]cyclopropyl}carbonyl)amino]ethyl}-1,1′-biphenyl-2-carboxylate (MK-0686), a Bradykinin B1 Receptor Antagonist

2008 Journal of Pharmacology and Experimental Therapeutics
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A General and Efficient 2-Amination of Pyridines and Quinolines.

2007 ChemInform
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Synthesis of [14C]tert‐butyl acetylene

2007 Journal of Labelled Compounds and Radiopharmaceuticals
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Synthesis of 2-Aminopyridines and 2-Amino-Quinolines from Their N-Oxides

2007 Synfacts
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Observations of Rhodium‐Containing Reaction Intermediates using HPLC with ICP‐MS and ESI‐MS Detection

2006 Advanced Synthesis & Catalysis
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Citations (20)