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Luca Canciani
Luca Canciani
Stereochemistry
Chemistry
Selectivity
Cytochrome P450
In vitro
3
Papers
22
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Discovery, synthesis, selectivity modulation and DMPK characterization of 5-azaspiro[2.4]heptanes as potent orexin receptor antagonists
2013
Bioorganic & Medicinal Chemistry Letters
Luigi Piero Stasi
Roberto Artusi
Clara Bovino
Benedetta Buzzi
Luca Canciani
Gianfranco Caselli
Fabrizio Colace
Paolo Garofalo
Silvia Giambuzzi
Patrice Larger
Ornella Letari
Stefano Mandelli
Lorenzo Perugini
Sabrina Pucci
Matteo Salvi
PierLuigi Toro
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Citations (10)
Synthesis, pharmacophore modeling and in vitro activity of 10,11-dihydrodibenzo[b,f]oxepine-4-carboxamide derivatives as novel and potent antagonists of the prostaglandin EP4 receptor.
2011
Bioorganic & Medicinal Chemistry Letters
Luigi Piero Stasi
Kanji Bhimani
Manuela Borriello
Luca Canciani
Gianfranco Caselli
Fabrizio Colace
Cristian Ferioli
Mehul Kaswala
Laura Mennuni
Tiziana Piepoli
Sabrina Pucci
Matteo Salvi
Vikas Shirsath
Tiziano Zanelli
Silvia Zerbi
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Citations (4)
In Vitro Study of the Inhibition and Induction of Human Cytochromes P450 by Crystalline Glucosamine Sulfate
2009
Drug metabolism and drug interactions
Stefano Persiani
Luca Canciani
Patrice Larger
Roberto Rotini
Giovanni Trisolino
Diego Antonioli
Lucio C. Rovati
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Citations (8)
1