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Fabrizio Colace
Fabrizio Colace
Chemistry
Selectivity
Cytochrome P450
Stereochemistry
Receptor
5
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38
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Compounds 4,4-difluoro-piperidine
2013
Luigi Piero Stasi
Lucio Claudio Rovati
Roberto Artusi
Clara Bovino
Fabrizio Colace
Stefano Mandelli
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Discovery, synthesis, selectivity modulation and DMPK characterization of 5-azaspiro[2.4]heptanes as potent orexin receptor antagonists
2013
Bioorganic & Medicinal Chemistry Letters
Luigi Piero Stasi
Roberto Artusi
Clara Bovino
Benedetta Buzzi
Luca Canciani
Gianfranco Caselli
Fabrizio Colace
Paolo Garofalo
Silvia Giambuzzi
Patrice Larger
Ornella Letari
Stefano Mandelli
Lorenzo Perugini
Sabrina Pucci
Matteo Salvi
PierLuigi Toro
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espiroamínicos compounds as orexin antogonistas
2012
Luigi Piero Stasi
Lucio Claudio Rovati
Roberto Artusi
Fabrizio Colace
Stefano Mandelli
Lorenzo Perugini
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Synthesis, pharmacophore modeling and in vitro activity of 10,11-dihydrodibenzo[b,f]oxepine-4-carboxamide derivatives as novel and potent antagonists of the prostaglandin EP4 receptor.
2011
Bioorganic & Medicinal Chemistry Letters
Luigi Piero Stasi
Kanji Bhimani
Manuela Borriello
Luca Canciani
Gianfranco Caselli
Fabrizio Colace
Cristian Ferioli
Mehul Kaswala
Laura Mennuni
Tiziana Piepoli
Sabrina Pucci
Matteo Salvi
Vikas Shirsath
Tiziano Zanelli
Silvia Zerbi
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Progress towards the identification of new aggrecanase inhibitors.
2009
Current Medicinal Chemistry
Francesca De Rienzo
Puneet Saxena
Federico Filomia
Gianfranco Caselli
Fabrizio Colace
Luigi Piero Stasi
Antonio Giordani
Maria Cristina Menziani
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Citations (24)
1