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Hidenobu Murafuji
Hidenobu Murafuji
Biochemistry
Kallikrein
Stratum corneum chymotryptic enzyme
KLK7
Chemistry
4
Papers
27
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Discovery and structure-activity relationship of imidazolinylindole derivatives as kallikrein 7 inhibitors.
2019
Bioorganic & Medicinal Chemistry Letters
Hidenobu Murafuji
Tsuyoshi Muto
Megumi Goto
Seiichi Imajo
Hajime Sugawara
Yoshiaki Oyama
Yutaka Minamitsuji
Shuji Miyazaki
Kenichi Murai
Hiromichi Fujioka
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Citations (6)
Structure-based drug design to overcome species differences in kallikrein 7 inhibition of 1,3,6-trisubstituted 1,4-diazepan-7-ones.
2018
Bioorganic & Medicinal Chemistry
Hidenobu Murafuji
Hajime Sugawara
Megumi Goto
Yoshiaki Oyama
Hiroki Sakai
Seiichi Imajo
Toshiyuki Tomoo
Tsuyoshi Muto
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Citations (5)
Structure-based drug design of 1,3,6-trisubstituted 1,4-diazepan-7-ones as selective human kallikrein 7 inhibitors
2018
Bioorganic & Medicinal Chemistry Letters
Hidenobu Murafuji
Hiroki Sakai
Megumi Goto
Yoshiaki Oyama
Seiichi Imajo
Hajime Sugawara
Toshiyuki Tomoo
Tsuyoshi Muto
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Citations (5)
Discovery and structure–activity relationship study of 1,3,6-trisubstituted 1,4-diazepane-7-ones as novel human kallikrein 7 inhibitors
2017
Bioorganic & Medicinal Chemistry Letters
Hidenobu Murafuji
Hiroki Sakai
Megumi Goto
Seiichi Imajo
Hajime Sugawara
Tsuyoshi Muto
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Citations (11)
1