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Tan Haizhong
Tan Haizhong
Biochemistry
cGMP-specific phosphodiesterase type 5
In vivo
Pharmacology
Chemistry
4
Papers
132
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Discovery of in Vivo Chemical Probes for Treating Alzheimer’s Disease: Dual Phosphodiesterase 5 (PDE5) and Class I Histone Deacetylase Selective Inhibitors
2019
ACS Chemical Neuroscience
Obdulia Rabal
Juan A. Sánchez-Arias
Mar Cuadrado-Tejedor
Irene de Miguel
Marta Pérez-González
Carolina García-Barroso
Ana Ugarte
Ander Estella-Hermoso de Mendoza
Elena Sáez
Maria Espelosin
Susana Ursua
Tan Haizhong
Wu Wei
Xu Musheng
Ana García-Osta
Julen Oyarzabal
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Citations (20)
Design, synthesis, biological evaluation and in vivo testing of dual phosphodiesterase 5 (PDE5) and histone deacetylase 6 (HDAC6)-selective inhibitors for the treatment of Alzheimer's disease
2018
European Journal of Medicinal Chemistry
Obdulia Rabal
Juan A. Sánchez-Arias
Mar Cuadrado-Tejedor
Irene de Miguel
Marta Pérez-González
Carolina García-Barroso
Ana Ugarte
Ander Estella-Hermoso de Mendoza
Elena Sáez
Maria Espelosin
Susana Ursua
Tan Haizhong
Wu Wei
Xu Musheng
Ana García-Osta
Julen Oyarzabal
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Citations (31)
Impact of Scaffold Exploration on Novel Dual-Acting Histone Deacetylases and Phosphodiesterase 5 Inhibitors for the Treatment of Alzheimer’s Disease
2017
ACS Chemical Neuroscience
Juan A. Sánchez-Arias
Obdulia Rabal
Mar Cuadrado-Tejedor
Irene de Miguel
Marta Pérez-González
Ana Ugarte
Elena Sáez
Maria Espelosin
Susana Ursua
Tan Haizhong
Wu Wei
Xu Musheng
Ana García-Osta
Julen Oyarzabal
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Citations (28)
Design, Synthesis, and Biological Evaluation of First-in-Class Dual Acting Histone Deacetylases (HDACs) and Phosphodiesterase 5 (PDE5) Inhibitors for the Treatment of Alzheimer’s Disease
2016
Journal of Medicinal Chemistry
Obdulia Rabal
Juan A. Sánchez-Arias
Mar Cuadrado-Tejedor
Irene de Miguel
Marta Pérez-González
Carolina García-Barroso
Ana Ugarte
Ander Estella-Hermoso de Mendoza
Elena Sáez
Maria Espelosin
Susana Ursua
Tan Haizhong
Wu Wei
Xu Musheng
Ana García-Osta
Julen Oyarzabal
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Citations (53)
1