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Emiliano Tamanini

Astex

11

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187

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Structure-Based Design of Potent and Orally Active Isoindolinone Inhibitors of MDM2-p53 Protein-Protein Interaction.

2021 Journal of Medicinal Chemistry
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Abstract 1652: Development of a potent class of small molecule inhibitors of the MDM2-p53 protein-protein interaction

2018 Cancer Research
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Preparation of isoindolinones as inhibitors of the MDM2-p53 interaction having anticancer activity

2017
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Discovery of a Potent Nonpeptidomimetic, Small-Molecule Antagonist of Cellular Inhibitor of Apoptosis Protein 1 (cIAP1) and X-Linked Inhibitor of Apoptosis Protein (XIAP).

2017 Journal of Medicinal Chemistry
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Structure of the Epigenetic Oncogene MMSET and Inhibition by N-Alkyl Sinefungin Derivatives

2016 ACS Chemical Biology
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Fragment-Based Discovery of Potent and Selective DDR1/2 Inhibitors

2015 ACS Medicinal Chemistry Letters
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Fragment-Based Drug Discovery Targeting Inhibitor of Apoptosis Proteins: Discovery of a Non-Alanine Lead Series with Dual Activity Against cIAP1 and XIAP.

2015 Journal of Medicinal Chemistry
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Abstract 2944: AT-IAP, a dual cIAP1 and XIAP antagonist with oral antitumor activity in melanoma models.

2013 Cancer Research
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Composés hétérocycliques bicycliques et leurs utilisations en thérapie

2012
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Abstract 2018: Discovery of potent dual inhibitors of both XIAP and cIAP1 using fragment based drug discovery

2012 Cancer Research
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