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Masahiro Sakaitani
Masahiro Sakaitani
Chugai Pharmaceutical Co.
In vivo
Chemistry
Biochemistry
Coumarin
Sulfamide
2
Papers
44
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The sulfamide moiety affords higher inhibitory activity and oral bioavailability to a series of coumarin dual selective RAF/MEK inhibitors.
2013
Bioorganic & Medicinal Chemistry Letters
Toshihiro Aoki
Ikumi Hyohdoh
Noriyuki Furuichi
Sawako Ozawa
Fumio Watanabe
Masayuki Matsushita
Masahiro Sakaitani
Kazutomo Ori
Kenji Takanashi
Naoki Harada
Yasushi Tomii
Mitsuyasu Tabo
Kiyoshi Yoshinari
Yuko Aoki
Nobuo Shimma
Hitoshi Iikura
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Citations (13)
Synthesis and structure-activity relationships of novel benzofuran farnesyltransferase inhibitors.
2009
Bioorganic & Medicinal Chemistry Letters
Kohsuke Asoh
Masami Kohchi
Ikumi Hyoudoh
Tatsuo Ohtsuka
Miyako Masubuchi
Kenichi Kawasaki
Hirosato Ebiike
Yasuhiko Shiratori
Takaaki A. Fukami
Osamu Kondoh
Toshiyuki Tsukaguchi
Nobuya Ishii
Yuko Aoki
Nobuo Shimma
Masahiro Sakaitani
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Citations (31)
1