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Jaroslava Paruchova
Jaroslava Paruchova
Schering-Plough
Biochemistry
Chemistry
Receptor
Melanin-concentrating hormone
Melanin-concentrating hormone receptor
4
Papers
167
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Bicyclic[4.1.0]heptanes as phenyl replacements for melanin concentrating hormone receptor antagonists.
2006
Bioorganic & Medicinal Chemistry
Ruo Xu
Shengjian Li
Jaroslava Paruchova
Mark D. McBriar
Henry Guzik
Anandan Palani
John W. Clader
Kathleen Cox
William J. Greenlee
Brian E. Hawes
Timothy J. Kowalski
Kim O’Neill
Brian Spar
Blair Weig
Daniel J. Weston
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Citations (21)
Discovery of orally efficacious melanin-concentrating hormone receptor-1 antagonists as antiobesity agents. Synthesis, SAR, and biological evaluation of bicyclo[3.1.0]hexyl ureas.
2006
Journal of Medicinal Chemistry
McBriar
Henry Guzik
Sherry Shapiro
Jaroslava Paruchova
Ruo Xu
Anandan Palani
John W. Clader
Kathleen Cox
William J. Greenlee
Brian E. Hawes
Timothy J. Kowalski
Kim O’Neill
Brian Spar
Blair Weig
Daniel J. Weston
Constance Farley
John Cook
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Citations (64)
Bicyclo[3.1.0]hexyl urea melanin concentrating hormone (MCH) receptor-1 antagonists : Impacting hERG liability via aryl modifications
2006
Bioorganic & Medicinal Chemistry Letters
Mark D. McBriar
Henry Guzik
Sherry Shapiro
Ruo Xu
Jaroslava Paruchova
John W. Clader
Kim O’Neill
Brian E. Hawes
Steve Sorota
Michael Margulis
Kristal Tucker
Daniel J. Weston
Kathleen Cox
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Citations (13)
Discovery of Bicycloalkyl Urea Melanin Concentrating Hormone Receptor Antagonists: Orally Efficacious Antiobesity Therapeutics
2005
Journal of Medicinal Chemistry
Mark D. McBriar
Henry Guzik
Ruo Xu
Jaroslava Paruchova
Shengjian Li
Anandan Palani
John W. Clader
William J. Greenlee
Brian E. Hawes
Timothy J. Kowalski
Kim O’Neill
Brian Spar
Blair Weig
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Citations (69)
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