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Robert A. Copeland
Robert A. Copeland
Bristol-Myers Squibb
Enzyme
Chemistry
Biochemistry
Substrate (chemistry)
Stereochemistry
5
Papers
113
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Beyond U0126. Dianion chemistry leading to the rapid synthesis of a series of potent MEK inhibitors
2004
Bioorganic & Medicinal Chemistry Letters
John Wityak
Frank W. Hobbs
Daniel S. Gardner
Joseph B. Santella
Joseph J. Petraitis
Jung Hui Sun
Margaret F. Favata
Andrea J. Daulerio
Kurumi Y. Horiuchi
Robert A. Copeland
Peggy A. Scherle
Bruce D. Jaffe
James M. Trzaskos
Ronald L. Magolda
George L. Trainor
John V. Duncia
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Citations (29)
Kinetic Studies on -Site Amyloid Precursor Protein-cleaving Enzyme (BACE)
2003
Larisa Toulokhonova
William J. Metzler
Mark R. Witmer
Robert A. Copeland
Jovita Marcinkeviciene
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Citations (2)
Kinetic Studies on β-Site Amyloid Precursor Protein-cleaving Enzyme (BACE) CONFIRMATION OF AN ISO-MECHANISM
2003
Journal of Biological Chemistry
Larisa Toulokhonova
William J. Metzler
Mark R. Witmer
Robert A. Copeland
Jovita Marcinkeviciene
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Citations (41)
A microplate assay specific for the enzyme aggrecanase.
2003
Analytical Biochemistry
Jeffery A Miller
Rui-Qin Liu
Gary L Davis
Michael Pratta
James M. Trzaskos
Robert A. Copeland
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Citations (26)
Novel Inhibition of Porcine Pepsin by a Substituted Piperidine PREFERENCE FOR ONE OF THE ENZYME CONFORMERS
2002
Journal of Biological Chemistry
Jovita Marcinkeviciene
Lisa M. Kopcho
Tao Yang
Robert A. Copeland
Brian M. Glass
Andrew P. Combs
Nikoo Falahatpisheh
Lorin A. Thompson
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Citations (15)
1