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Simone V. Bigi
Simone V. Bigi
Takeda Pharmaceutical Company
Biochemistry
Chemistry
Mitogen-activated protein kinase kinase
ASK1
Mitogen-activated protein kinase
2
Papers
50
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Discovery of 7-Oxo-2,4,5,7-tetrahydro-6H-pyrazolo[3,4-c]pyridine Derivatives as Potent, Orally Available, and Brain-penetrating Receptor Interacting Protein 1 (RIP1) Kinase Inhibitors; Analysis of Structure–Kinetic Relationships
2018
Journal of Medicinal Chemistry
Masato Yoshikawa
Morihisa Saitoh
Taisuke Katoh
Tomohiro Seki
Simone V. Bigi
Yuji Shimizu
Tsuyoshi Ishii
Takuro Okai
Masako Kuno
Harumi Hattori
Etsuro Watanabe
Kumar Singh Saikatendu
Hua Zou
Masanori Nakakariya
Takayuki Tatamiya
Yoshihisa Nakada
Takatoshi Yogo
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Fragment-based drug discovery of potent and selective MKK3/6 inhibitors.
2016
Bioorganic & Medicinal Chemistry Letters
Mark E. Adams
Toshitake Kobayashi
J. David Lawson
Morihisa Saitoh
Kenichiro Shimokawa
Simone V. Bigi
Mark S. Hixon
Christopher Smith
Takayuki Tatamiya
Masayuki Goto
Joseph Russo
Charles E. Grimshaw
Steven Swann
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Citations (13)
1