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E.C. Breinlinger
E.C. Breinlinger
Stereochemistry
Chemistry
Crystal structure
Inverse agonist
Triazole
3
Papers
18
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Crystal structure of human ROR gamma LBD in complex with a (quinolinoxymethyl)benzamide inverse agonist
2020
J. Amaudrut
M.A. Argiriadi
M. Barth
E.C. Breinlinger
D.J. Calderwood
K.P. Cusack
M.E. Kort
C. Montalbetti
D. Potin
O. Poupardin
L. Spitzer
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Crystal structure of human ROR gamma LBD in complex with a quinoline sulfonamide inverse agonist
2019
F Ciesielski
J. Amaudrut
M.A. Argiriadi
M. Barth
E.C. Breinlinger
D.J. Calderwood
K.P. Cusack
M.E. Kort
C. Montalbetti
D. Potin
O. Poupardin
L. Spitzer
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Structure-based design and subsequent optimization of 2-tolyl-(1,2,3-triazol-1-yl-4-carboxamide) inhibitors of p38 MAP kinase
2008
Bioorganic & Medicinal Chemistry Letters
Derek Cogan
Ronald A. Aungst
E.C. Breinlinger
Tazmeen N. Fadra
Daniel R. Goldberg
Ming-Hong Hao
Rachel R. Kroe
Neil Moss
Christopher Pargellis
Kevin Chungeng Qian
Alan David Swinamer
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Citations (18)
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