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T. Yoon
T. Yoon
Novartis
Stereochemistry
Complement Factor D
Chemistry
Fragment-based lead discovery
Biology
4
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4
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Complement factor D in complex with the inhibitor 3-((3-((3-(aminomethyl)phenyl)amino)-1H-pyrazolo[3,4-d]pyrimidin-4-yl)amino)phenol
2018
A. Mac Sweeney
Nils Ostermann
Anna Vulpetti
Jürgen Maibaum
P. Erbel
Edwige Liliane Jeanne Lorthiois
T. Yoon
Stefan Andreas Randl
Simon Ruedisser
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Complement factor D in complex with the inhibitor (4-((3-(aminomethyl)phenyl)amino)quinazolin-2-yl)-L-valine
2018
A. Mac Sweeney
Nils Ostermann
Anna Vulpetti
Jürgen Maibaum
P. Erbel
Edwige Liliane Jeanne Lorthiois
T. Yoon
Stefan Andreas Randl
Simon Ruedisser
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Complement factor D in complex with the inhibitor N-(3'-(aminomethyl)-[1,1'-biphenyl]-3-yl)-3-methylbutanamide
2018
A. Mac Sweeney
Nils Ostermann
Anna Vulpetti
Jürgen Maibaum
P. Erbel
Edwige Liliane Jeanne Lorthiois
T. Yoon
Stefan Andreas Randl
Simon Ruedisser
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Discovery and Design of First Benzylamine-Based Ligands Binding to an Unlocked Conformation of the Complement Factor D.
2018
ACS Medicinal Chemistry Letters
Anna Vulpetti
Nils Ostermann
Stefan Andreas Randl
T. Yoon
A. Mac Sweeney
Frederic Cumin
Edwige Liliane Jeanne Lorthiois
Simon Rüdisser
P. Erbel
Jürgen Maibaum
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Citations (4)
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