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Takahiro Kitamura
Takahiro Kitamura
Daiichi Sankyo
Chemistry
Antibacterial activity
Biochemistry
Stereochemistry
Quinolone
4
Papers
47
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Discovery of Novel 7-[(1 R ,5 S )-1-Amino-5-fluoro-3-azabicyclo[3.3.0]octan-3-yl]-6-fluoro-1-[(1 R ,2 S )-2-fluorocyclopropane]-8-(methoxy or methyl)quinolones
2019
Chemical & Pharmaceutical Bulletin
Satoshi Komoriya
Takashi Odagiri
Hiroaki Inagaki
Masatoshi Nagamochi
Rie Miyauchi
Ken-ichi Yoshida
Takahiro Kitamura
Hisashi Takahashi
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Citations (2)
Design, Synthesis, and Biological Evaluation of Novel 7-[(3aS,7aS)-3a-Aminohexahydropyrano[3,4-c]pyrrol-2(3H)-yl]-8-methoxyquinolines with Potent Antibacterial Activity against Respiratory Pathogens
2018
Journal of Medicinal Chemistry
Takashi Odagiri
Hiroaki Inagaki
Masatoshi Nagamochi
Takahiro Kitamura
Satoshi Komoriya
Hisashi Takahashi
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Citations (7)
Discovery and structure-guided fragment-linking of 4-(2,3-dichlorobenzoyl)-1-methyl-pyrrole-2-carboxamide as a pyruvate kinase M2 activator
2017
Bioorganic & Medicinal Chemistry
Yumi Matsui
Isao Yasumatsu
Takashi Asahi
Takahiro Kitamura
Kazuo Kanai
Osamu Ubukata
Hitoshi Hayasaka
Sachiko Takaishi
Hiroyuki Hanzawa
Shin‐ichi Katakura
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Citations (15)
Design, synthesis, and biological evaluations of novel 7-[7-amino-7-methyl-5-azaspiro[2.4]heptan-5-yl]-8-methoxyquinolines with potent antibacterial activity against respiratory pathogens.
2013
Journal of Medicinal Chemistry
Takashi Odagiri
Hiroaki Inagaki
Yuichi Sugimoto
Masatoshi Nagamochi
Rie N. Miyauchi
Junichi Kuroyanagi
Takahiro Kitamura
Satoshi Komoriya
Hisashi Takahashi
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Citations (23)
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