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Anthony D. Garcia
Anthony D. Garcia
École Normale Supérieure
Chemistry
Stereochemistry
Biochemistry
KEAP1
Derivatization
3
Papers
47
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Deconstructing Noncovalent Kelch-like ECH-Associated Protein 1 (Keap1) Inhibitors into Fragments to Reconstruct New Potent Compounds.
2021
Journal of Medicinal Chemistry
Jakob S. Pallesen
Dilip Narayanan
Kim T. Tran
Sara Marie Øie Solbak
Giuseppe Marseglia
Louis M.E. Sørensen
Lars Jakobsen Høj
Federico Munafò
Rosa M. C. Carmona
Anthony D. Garcia
Haritha L. Desu
Roberta Brambilla
Tommy N. Johansen
Grzegorz M. Popowicz
Michael Sattler
Michael Gajhede
Anders Bach
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Citations (5)
Synthesis, Derivatization, and Structural Analysis of Phosphorylated Mono-, Di-, and Trifluorinated d-Gluco-heptuloses by Glucokinase: Tunable Phosphoglucomutase Inhibition
2019
Jian-She Zhu
Kyle M. Stiers
Sherany M. Winter
Anthony D. Garcia
Antoine F. Versini
L.J. Beamer
David L. Jakeman
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Citations (6)
A Comparative AssessmentStudy of Known Small-MoleculeKeap1−Nrf2 Protein–Protein Interaction Inhibitors: ChemicalSynthesis, Binding Properties, and Cellular Activity
2019
Journal of Medicinal Chemistry
Kim T. Tran
Jakob S. Pallesen
Sara Marie Øie Solbak
Dilip Narayanan
Amina Baig
Jie Zang
Alejandro Aguayo-Orozco
Rosa M. C. Carmona
Anthony D. Garcia
Anders Bach
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Citations (36)
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