author-photo

Anna S. Gardberg

Emerald Group Publishing

31

Papers

512

Citations

Citation Trend

Filter By

Papers (17) Sort By

Journal Conference Others

Discovery of CPI-1612: A Potent, Selective, and Orally Bioavailable EP300/CBP Histone Acetyltransferase (HAT) Inhibitor

2020 ACS Medicinal Chemistry Letters
Show All
- Source
- Cite
- Save
Citations (15)
Optimization of the efflux ratio and permeability of covalent irreversible BTK inhibitors

2018 Bioorganic & Medicinal Chemistry Letters
Show All
- Source
- Cite
- Save
Citations (5)
Discovery of a novel series of pyridine and pyrimidine carboxamides as potent and selective covalent inhibitors of Btk

2018 Bioorganic & Medicinal Chemistry Letters
Show All
- Source
- Cite
- Save
Citations (9)
Discovery of potent, highly selective covalent irreversible BTK inhibitors from a fragment hit.

2018 Bioorganic & Medicinal Chemistry Letters
Show All
- Source
- Cite
- Save
Citations (13)
Ability of Bruton's Tyrosine Kinase Inhibitors to Sequester Y551 and Prevent Phosphorylation Determines Potency for Inhibition of Fc Receptor but not B-Cell Receptor Signaling.

2017 Molecular Pharmacology
Show All
- Source
- Cite
- Save
Citations (59)
Increasing the structural coverage of tuberculosis drug targets.

2015 Tuberculosis
Show All
- Source
- Cite
- Save
Citations (79)
Structure of uridine diphosphate N-acetylglucosamine pyrophosphorylase from Entamoeba histolytica

2015 Acta Crystallographica Section F-structural Biology and Crystallization Communications
Show All
- Source
- Cite
- Save
Citations (0)
Structural basis for the inhibition of poly(ADP-ribose) polymerases 1 and 2 by BMN 673, a potent inhibitor derived from dihydropyridophthalazinone.

2014 Acta Crystallographica Section F-structural Biology and Crystallization Communications
Show All
- Source
- Cite
- Save
Citations (31)
Composés hétéroaryle servant d'inhibiteurs de la btk et leurs utilisations

2014
Show All
- Source
- Cite
- Save
Citations (0)
Structural Insights into the Functional Role of the Hcn Sub-domain of the Receptor-Binding Domain of the Botulinum Neurotoxin Mosaic Serotype C/D

2013 Biochimie
Show All
- Source
- Cite
- Save
Citations (8)