Screening of benzenesulfonamide in combination with chemically diverse fragments against carbonic anhydrase by differential scanning fluorimetry

Mikhail Krasavin,Stanislav Kalinin,Sergey Zozulya,Anastasiia Gryniukova,Petro Borysko,Andrea Angeli,Claudiu T. Supuran

Screening of benzenesulfonamide in combination with chemically diverse fragments against carbonic anhydrase by differential scanning fluorimetry

2020

Mikhail Krasavin
Stanislav Kalinin
Sergey Zozulya
Anastasiia Gryniukova
Petro Borysko
Andrea Angeli
Claudiu T. Supuran

AbstractThe differential scanning fluorimetry (DSF) screening of 5.692 fragments in combination with benzenesulfonamide (BSA) against bovine carbonic anhydrase (bCA) delivered >100 hits that either...

Keywords:

Chemistry
Carbonic anhydrase
Biochemistry
Fluorescence spectroscopy
Thermal shift assay
Fragment-based lead discovery
Carbonic anhydrase II

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