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Federico Da Settimo

University of Pisa

174

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3248

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Allosterism vs. Orthosterism: Recent Findings and Future Perspectives on A2B AR Physio-Pathological Implications

2021 Frontiers in Pharmacology
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De novo Neurosteroidogenesis in Human Microglia: Involvement of the 18 kDa Translocator Protein.

2021 International Journal of Molecular Sciences
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The Alpha Keto Amide Moiety as a Privileged Motif in Medicinal Chemistry: Current Insights and Emerging Opportunities

2021 Journal of Medicinal Chemistry
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Carbonic anhydrase activation profile of indole-based derivatives.

2021 Journal of Enzyme Inhibition and Medicinal Chemistry
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Synthesis and Screening in Mice of Fluorine-Containing PET Radioligands for TSPO: Discovery of a Promising 18F-Labeled Ligand.

2021 Journal of Medicinal Chemistry
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Tetrahydroquinazole-based secondary sulphonamides as carbonic anhydrase inhibitors: synthesis, biological evaluation against isoforms I, II, IV, and IX, and computational studies

2021 Journal of Enzyme Inhibition and Medicinal Chemistry
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Novel positive allosteric modulators of A2B adenosine receptor acting as bone mineralisation promoters.

2021 Journal of Enzyme Inhibition and Medicinal Chemistry
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Inhibition studies on carbonic anhydrase isoforms I, II, IV and IX with N-arylsubstituted secondary sulfonamides featuring a bicyclic tetrahydroindazole scaffold.

2021 European Journal of Medicinal Chemistry
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Exploiting the Indole Scaffold to Design Compounds Binding to Different Pharmacological Targets.

2020 Molecules
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Targeting the KRAS Oncogene: Synthesis, Physicochemical and Biological Evaluation of Novel G-Quadruplex DNA Binders.

2020 European Journal of Pharmaceutical Sciences
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