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Nicola Porta
Nicola Porta
University of Padua
Pyrimidine
Adenosine receptor
Chemistry
Stereochemistry
Biochemistry
3
Papers
47
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5,7-Disubstituted-[1,2,4]triazolo[1,5-a][1,3,5]triazines as pharmacological tools to explore the antagonist selectivity profiles toward adenosine receptors
2016
European Journal of Medicinal Chemistry
Stephanie Federico
Antonella Ciancetta
Nicola Porta
Sara Redenti
Giorgia Pastorin
Barbara Cacciari
Karl-Norbert Klotz
Stefano Moro
Giampiero Spalluto
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Citations (14)
7-Amino-2-phenylpyrazolo[4,3-d]pyrimidine derivatives: Structural investigations at the 5-position to target human A1 and A2A adenosine receptors. Molecular modeling and pharmacological studies
2014
European Journal of Medicinal Chemistry
Lucia Squarcialupi
Vittoria Colotta
Daniela Catarzi
Flavia Varano
Marco Betti
Katia Varani
Fabrizio Vincenzi
Pier Andrea Borea
Nicola Porta
Antonella Ciancetta
Stefano Moro
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Citations (22)
Scaffold decoration at positions 5 and 8 of 1,2,4-triazolo[1,5-c]pyrimidines to explore the antagonist profiling on adenosine receptors: a preliminary structure-activity relationship study.
2014
Journal of Medicinal Chemistry
Stephanie Federico
Antonella Ciancetta
Nicola Porta
Sara Redenti
Giorgia Pastorin
Barbara Cacciari
Karl-Norbert Klotz
Stefano Moro
Giampiero Spalluto
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Citations (11)
1