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Naga Rajiv Lakkaniga
Naga Rajiv Lakkaniga
Scripps Research Institute
Chemistry
Mutation
Mutant
Kinase
Protein kinase domain
2
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2024
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Discovery of imidazo[1,2-a]pyridine-thiophene derivatives as FLT3 and FLT3 mutants inhibitors for acute myeloid leukemia through structure-based optimization of an NEK2 inhibitor.
2021
European Journal of Medicinal Chemistry
Lingtian Zhang
Naga Rajiv Lakkaniga
Jaideep B. Bharate
Nicholas Mcconnell
Xiuqi Wang
Anupreet Kharbanda
Yuet-Kin Leung
Brendan Frett
Neil P. Shah
Hong Yu Li
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Novel hydroxybenzylamine-deoxyvasicinone hybrids as anticholinesterase therapeutics for Alzheimer's disease.
2021
Bioorganic & Medicinal Chemistry
Suresh K. Bowroju
Narsimha Reddy Penthala
Naga Rajiv Lakkaniga
Meenakshisundaram Balasubramaniam
Srinivas Ayyadevara
Robert J. Shmookler Reis
Peter A. Crooks
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