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Thaddeus Tomaszek
Thaddeus Tomaszek
GlaxoSmithKline
Biochemistry
Chemistry
Stereochemistry
Enzyme
Nitrile
3
Papers
29
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Discovery of renin inhibitors containing a simple aspartate binding moiety that imparts reduced P450 inhibition.
2017
Bioorganic & Medicinal Chemistry Letters
Brian G. Lawhorn
Tritin Tran
Victor S. Hong
Lisa Morgan
BaoChau T. Le
Mark R. Harpel
Larry J. Jolivette
Elsie Diaz
Benjamin Schwartz
Jeffrey W. Gross
Thaddeus Tomaszek
Simon F. Semus
Nestor O. Concha
Angela Smallwood
Dennis A. Holt
Lara S. Kallander
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2-Cyano-4-fluoro-1-thiovalylpyrrolidine analogues as potent inhibitors of DPP-IV
2005
Bioorganic & Medicinal Chemistry Letters
Curt D. Haffner
Darryl L. McDougald
Steven Michael Reister
Brian Thompson
Christopher R. Conlee
Jing Fang
Jonathan Y. Bass
James M. Lenhard
Dallas K. Croom
Melissa B. Secosky-Chang
Thaddeus Tomaszek
Donavon McConn
Kevin J. Wells-Knecht
Paul R. Johnson
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Citations (20)
1