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Arnaud Descours
Arnaud Descours
Pfizer
Enzyme
Biochemistry
Organic chemistry
Chemical synthesis
Stereochemistry
3
Papers
92
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Spiroquinazolinones as novel, potent, and selective PDE7 inhibitors. Part 1
2004
Bioorganic & Medicinal Chemistry Letters
Edwige Lorthiois
Patrick Bernardelli
Fabrice Vergne
Chrystelle Oliveira
Abdel-Kader Mafroud
Emmanuelle Proust
Lamia Heuze
François Moreau
Moulay Idrissi
Anita Tertre
Bernadette Bertin
Magali Coupe
Roger Wrigglesworth
Arnaud Descours
Patricia Soulard
Patrick Berna
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Citations (33)
Discovery of thiadiazoles as a novel structural class of potent and selective PDE7 inhibitors. Part 2: Metabolism-directed optimization studies towards orally bioavailable derivatives
2004
Bioorganic & Medicinal Chemistry Letters
Fabrice Vergne
Patrick Bernardelli
Edwige Lorthiois
Nga Pham
Emmanuelle Proust
Chrystelle Oliveira
Abdel-Kader Mafroud
Pierre Ducrot
Roger Wrigglesworth
Françoise Berlioz-Seux
Francis Coleon
Eric Chevalier
François Moreau
Moulay Idrissi
Anita Tertre
Arnaud Descours
Patrick Berna
Mei Li
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Citations (33)
Spiroquinazolinones as novel, potent, and selective PDE7 inhibitors. Part 2: Optimization of 5,8-disubstituted derivatives
2004
Bioorganic & Medicinal Chemistry Letters
Patrick Bernardelli
Edwige Lorthiois
Fabrice Vergne
Chrystelle Oliveira
Abdel-Kader Mafroud
Emmanuelle Proust
Nga Pham
Pierre Ducrot
François Moreau
Moulay Idrissi
Anita Tertre
Bernadette Bertin
Magali Coupe
Eric Chevalier
Arnaud Descours
Françoise Berlioz-Seux
Patrick Berna
Mei Li
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Citations (26)
1