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Simon Gonzalez
Simon Gonzalez
Vrije Universiteit Brussel
Chemistry
Pharmacology
Neurotensin
Receptor
Ligand
3
Papers
16
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Optimized Opioid-Neurotensin Multitarget Peptides: From Design to Structure-Activity Relationship Studies.
2020
Journal of Medicinal Chemistry
Simon Gonzalez
Maria Dumitrascuta
Emilie Eiselt
Stevany Louis
Linda Kunze
Annalisa Blasiol
Mélanie Vivancos
Santo Previti
Elke Dewolf
Charlotte Martin
Dirk Tourwé
Florine Cavelier
Louis Gendron
Philippe Sarret
Mariana Spetea
Steven Ballet
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Citations (3)
Structure-Based Design of Melanocortin 4 Receptor Ligands Based on the SHU-9119-hMC4R Cocrystal Structure†.
2020
Journal of Medicinal Chemistry
Charlotte Martin
Luis E. Gimenez
Savannah Y. Williams
Yu Jing
Yiran Wu
Charlie Hollanders
Olivier Van der Poorten
Simon Gonzalez
Kevin Van holsbeeck
Santo Previti
Arthur Lamouroux
Suwen Zhao
Dirk Tourwé
Raymond C. Stevens
Roger D. Cone
Steven Ballet
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Citations (2)
Neurotensin Analogues Containing Cyclic Surrogates of Tyrosine at Position 11 Improve NTS2 Selectivity Leading to Analgesia without Hypotension and Hypothermia
2019
ACS Chemical Neuroscience
Emilie Eiselt
Simon Gonzalez
Charlotte Martin
Magali Chartier
Cecilia Betti
Jean-Michel Longpré
Florine Cavelier
Dirk Tourwé
Louis Gendron
Steven Ballet
Philippe Sarret
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Citations (11)
1