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Tetsuyoshi Matsufuji
Tetsuyoshi Matsufuji
Daiichi Sankyo
Chemistry
Biochemistry
Stereochemistry
In vivo
Fatty acid
5
Papers
49
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Synthesis and biological evaluation of novel chiral diazepine derivatives as bombesin receptor subtype-3 (BRS-3) agonists incorporating an antedrug approach.
2015
Bioorganic & Medicinal Chemistry
Tetsuyoshi Matsufuji
Kousei Shimada
Shozo Kobayashi
Masanori Ichikawa
Asuka Kawamura
Teppei Fujimoto
Tsuyoshi Arita
Takashi Hara
Masahiro Konishi
Rie Abe-Ohya
Masanori Izumi
Yoshitaka Sogawa
Yoko Nagai
Kazuhiro Yoshida
Yasuyuki Abe
Takako Kimura
Hisashi Takahashi
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Citations (14)
Discovery of novel chiral diazepines as bombesin receptor subtype-3 (BRS-3) agonists with low brain penetration.
2014
Bioorganic & Medicinal Chemistry Letters
Tetsuyoshi Matsufuji
Kousei Shimada
Shozo Kobayashi
Asuka Kawamura
Teppei Fujimoto
Tsuyoshi Arita
Takashi Hara
Masahiro Konishi
Rie Abe-Ohya
Masanori Izumi
Yoshitaka Sogawa
Youko Nagai
Kazuhiro Yoshida
Hisashi Takahashi
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Citations (13)
Arylpiperazines as fatty acid transport protein 1 (FATP1) inhibitors with improved potency and pharmacokinetic properties.
2013
Bioorganic & Medicinal Chemistry Letters
Tetsuyoshi Matsufuji
Mika Ikeda
Asuka Naito
Masakazu Hirouchi
Shoichi Kanda
Masanori Izumi
Jun Harada
Tsuyoshi Shinozuka
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Citations (13)
Discovery and optimization of novel fatty acid transport protein 1 (FATP1) inhibitors.
2012
Bioorganic & Medicinal Chemistry Letters
Tetsuyoshi Matsufuji
Mika Ikeda
Asuka Naito
Masakazu Hirouchi
Hideo Takakusa
Shoichi Kanda
Masanori Izumi
Jun Harada
Tsuyoshi Shinozuka
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Citations (9)
Nouveau dérivé de phénylpyrrole
2009
Akihiro Furukawa
Takehiro Fukuzaki
Yukari Onishi
Hideki Kobayashi
Takeshi Honda
Yumi Matsui
Masahiro Konishi
Kenjiro Ueda
Tetsuyoshi Matsufuji
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