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Kenneth M. Gigstad

Millennium Pharmaceuticals

5

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214

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Identification of Novel Carbocyclic Pyrimidine Cyclic Dinucleotide STING Agonists for Antitumor Immunotherapy Using Systemic Intravenous Route.

2021 Journal of Medicinal Chemistry
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N,C-Capped Dipeptides with Selectivity for Mycobacterial Proteasome over Human Proteasomes: Role of S3 and S1 Binding Pockets

2013 Journal of the American Chemical Society
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Characterization of a new series of non-covalent proteasome inhibitors with exquisite potency and selectivity for the 20S β5-subunit

2010 Biochemical Journal
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Optimization of a series of dipeptides with a P3 threonine residue as non-covalent inhibitors of the chymotrypsin-like activity of the human 20S proteasome.

2010 Bioorganic & Medicinal Chemistry Letters
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