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Tsukasa Hasegawa
Tsukasa Hasegawa
University of Tokyo
Biochemistry
Kinase
Chemistry
Structure–activity relationship
Cell culture
3
Papers
17
Citations
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Design and Synthesis of Potent and Selective PIM Kinase Inhibitors by Targeting Unique Structure of ATP-Binding Pocket
2017
ACS Medicinal Chemistry Letters
Hirofumi Nakano
Tsukasa Hasegawa
Hirotatsu Kojima
Takayoshi Okabe
Tetsuo Nagano
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Citations (10)
Development of a potent and selective FLT3 kinase inhibitor by systematic expansion of a non-selective fragment-screening hit.
2016
Bioorganic & Medicinal Chemistry Letters
Hirofumi Nakano
Tsukasa Hasegawa
Riyo Imamura
Nae Saito
Hirotatsu Kojima
Takayoshi Okabe
Tetsuo Nagano
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Citations (4)
Design and synthesis of an in vivo-efficacious PIM3 kinase inhibitor as a candidate anti-pancreatic cancer agent
2015
Bioorganic & Medicinal Chemistry Letters
Hirofumi Nakano
Tsukasa Hasegawa
Nae Saito
Kaoru Furukawa
Naofumi Mukaida
Hirotatsu Kojima
Takayoshi Okabe
Tetsuo Nagano
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Citations (3)
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