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Conner Craigon
Conner Craigon
University of Dundee
Chemistry
protein degradation
Cooperativity
Ternary complex
Target protein
4
Papers
6
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0
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Mechanistic and Structural Features of PROTAC Ternary Complexes.
2021
Methods of Molecular Biology
Ryan Casement
Adam Bond
Conner Craigon
Alessio Ciulli
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Citations (2)
Trivalent PROTACs enhance protein degradation via combined avidity and cooperativity.
2021
Nature Chemical Biology
Satomi Imaide
Kristin M. Riching
Nikolai Makukhin
Vesna Vetma
Claire Whitworth
Scott J. Hughes
Nicole Trainor
Sarah D. Mahan
Nancy Murphy
Angus D Cowan
Kwok-Ho Chan
Conner Craigon
Andrea Testa
Chiara Maniaci
Marjeta Urh
Danette L. Daniels
Alessio Ciulli
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Citations (3)
Development of BromoTag: A "Bump-and-Hole"-PROTAC System to Induce Potent, Rapid, and Selective Degradation of Tagged Target Proteins.
2021
Journal of Medicinal Chemistry
Adam G. Bond
Conner Craigon
Kwok-Ho Chan
Andrea Testa
Athanasios Karapetsas
Rotimi Fasimoye
Thomas Macartney
J. Julian Blow
Dario R. Alessi
Alessio Ciulli
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Amide-to-ester substitution as a strategy for optimizing PROTAC permeability and cellular activity
2021
ChemRxiv
Victoria G. Klein
Adam Bond
Conner Craigon
R. Scott Lokey
Alessio Ciulli
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Citations (1)
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