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Jay Thomas Afragola
Jay Thomas Afragola
Chemistry
Organic chemistry
Stereochemistry
Biochemistry
Chirality (chemistry)
5
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175
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First Scale-Up Synthesis of WAY-262398, a Novel, Dual-Acting SSRI/5HT1a Antagonist
2009
Organic Process Research & Development
Antonia Nikitenko
Asaf Alimardanov
Jay Thomas Afragola
Jean Schmid
Livia Kristofova
Deborah Ann Evrard
Nicole T. Hatzenbuhler
Vasilios Marathias
Gary Paul Stack
Steve Lenicek
John R. Potoski
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Citations (8)
Practical Asymmetric Synthesis of Trifluoromethyl-Containing Aminoester Using a Modified Davis Protocol
2008
Organic Process Research & Development
Asaf Alimardanov
Jean Schmid
Jay Thomas Afragola
Gulnaz Khafizova
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Citations (9)
Synthesis and SAR of [1,2,4]triazolo[1,5-a]pyrimidines, a class of anticancer agents with a unique mechanism of tubulin inhibition.
2007
Journal of Medicinal Chemistry
Nan Zhang
Semiramis Ayral-Kaloustian
Thai Hiep Nguyen
Jay Thomas Afragola
Richard Hernandez
Judy Lucas
James Joseph Gibbons
Carl Beyer
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Citations (158)
4-(2,4-dichloro-5-methoxyphenyl)amino-6-methoxy-7-{[5-(amino substitue)methyl]-3-furyl}-3-quinolinecarbonitriles utilises en tant qu'inhibiteurs de kinase
2005
Jay Thomas Afragola
Asaf Alimardanov
Diane Harris Boschelli
Biqi Wu
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A process for the preparation of tubulinininhibitorer
2004
Semiramis Ayral-Kaloustian
Yanzhong Wu
Jean Schmid
Jay Thomas Afragola
David Michael Blum
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